- Chemicals, Inhibitors, Activators, Antagonists, and Agonists
ACALABRUTINIB (ACP196)
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AC220 (QUIZARTINIB)
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AMG-511
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AVL-292 (SPEBRUTINIB)
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TAK-981
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LYC-55716 (CINTIRORGON)
Cintirorgon (CAS No.: 2055536-64-4), is a first-in-class, selective and orally bioavailable RORγ agonist. Cintirorgon (LYC-55716) modulates gene expression of RORγ expressing T lymphocyte immune cells, resulting in enhanced effector…
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Darovasertib (LXS-196, NVP-LXS196, IDE196)
Darovasertib (CAS No.: 1874276-76-2), is a potent, selective and orally active protein kinase C (PKC) inhibitor, with IC50 values of 1.9 nM, 0.4 nM and 3.1 μM for PKCα,…
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ARQ-197
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M-3258 (M3258, M 3258)
M-3258 (CAS No.: 2285330-15-4), orally bioavailable, potent, reversible and highly selective immunoproteasome subunit LMP7 (β5i) inhibitor. M3258 exerts high biochemical (IC50=3.6 nM) and cellular (IC50=3.4 nM) potency against the…
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AMG-176
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