GSK046 (GSK-046, IBET-BD2)


GSK046 (iBET-BD2, GSK 046, GSK-046) (CAS No.: 2474876-09-8), a potent, selective and orally active BD2 bromodomain inhibitor of the BET proteins, with IC50s of 264 nM (BRD2 BD2), 98 nM (BRD3 BD2), 49 nM (BRD4 BD2) and 214 nM (BRDT BD2), respectively. >99% Purity.

Synonyms: iBET-BD2, GSK 046, GSK-046, BET Proteins, BRDT, BRD2, BRD3, BRD4

For Research Use Only.

SKU: APIM050401
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